Discovery and SAR of novel pyrazolo[1,5-a]pyrimidines as inhibitors of CDK9

Phillipson, Louisa J., Segal, David H., Nero, Tracy L., Parker, Michael W., Wan, Soo San, de Silva, Melanie, Guthridge, Mark A., Wei, AH and Burns, Christopher J. 2015, Discovery and SAR of novel pyrazolo[1,5-a]pyrimidines as inhibitors of CDK9, Bioorganic & medicinal chemistry, vol. 23, no. 19, pp. 6280-6296, doi: 10.1016/j.bmc.2015.08.035.

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Title Discovery and SAR of novel pyrazolo[1,5-a]pyrimidines as inhibitors of CDK9
Author(s) Phillipson, Louisa J.
Segal, David H.
Nero, Tracy L.
Parker, Michael W.
Wan, Soo San
de Silva, Melanie
Guthridge, Mark A.ORCID iD for Guthridge, Mark A. orcid.org/0000-0002-0536-3471
Wei, AH
Burns, Christopher J.
Journal name Bioorganic & medicinal chemistry
Volume number 23
Issue number 19
Start page 6280
End page 6296
Total pages 17
Publisher Elsevier
Place of publication Amsterdam, The Netherlands
Publication date 2015-10-01
ISSN 0968-0896
Keyword(s) CDK7
CDK9 selectivity
FLT3
Molecular modelling
PI3Kα
Pyrazolo[1,5-a]pyrimidine
Language eng
DOI 10.1016/j.bmc.2015.08.035
Indigenous content off
Field of Research 0304 Medicinal and Biomolecular Chemistry
1115 Pharmacology and Pharmaceutical Sciences
0305 Organic Chemistry
HERDC Research category C1 Refereed article in a scholarly journal
Persistent URL http://hdl.handle.net/10536/DRO/DU:30132334

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