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Structure activity refinement of phenylsulfonyl piperazines as antimalarials that block erythrocytic invasion
journal contribution
posted on 2021-03-15, 00:00 authored by W Nguyen, M G Dans, A Ngo, M R Gancheva, O Romeo, S Duffy, Tania De Koning-WardTania De Koning-Ward, K N Lowes, H J Sabroux, V M Avery, D W Wilson, P R Gilson, B E SleebsStructure activity refinement of phenylsulfonyl piperazines as antimalarials that block erythrocytic invasion
History
Journal
European journal of medicinal chemistryVolume
214Article number
113253Pagination
1 - 27Publisher
ElsevierLocation
Amsterdam, The NetherlandsPublisher DOI
ISSN
0223-5234eISSN
1768-3254Language
EnglishPublication classification
C1 Refereed article in a scholarly journalUsage metrics
Keywords
AntimalarialChemistry, MedicinalErythrocyte invasionLife Sciences & BiomedicineMalariaPharmacology & PharmacyPhenylsulfonyl piperazinePlasmodiumScience & TechnologyPLASMODIUM-FALCIPARUMARTEMISININ RESISTANCEMICROSOMAL METABOLISMMALARIA PARASITESCROSS-RESISTANCEBLOOD-STAGEINHIBITORSDRUGSIDENTIFICATIONGAMETOCYTESOrganic Chemistry
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